| 4EKC_A_B | SB179D | Guanine nucleotide-binding protein G(q) subunit alpha | Regulator of G-protein signaling 2 | 23434405 | IC50=0.27 ± 0.06 uM
LogEC50 (n)=2.1 ± 0.03 nM (20) | IC50=16.0 ± 4 uM
Log EC50 (n)=3.8 ± 0.26 nM (3) | flow-cytometry-based assay，25°C |
| 4EKC_A_B | SB179K | Guanine nucleotide-binding protein G(q) subunit alpha | Regulator of G-protein signaling 2 | 23434405 | IC50=0.27 ± 0.06 uM
LogEC50 (n)=2.1 ± 0.03 nM (20) | IC50=3.4 ± 0.9 uM
Log EC50 (n)=3.0 ± 0.07 nM (5) | flow-cytometry-based assay，25°C |
| 4EKC_A_B | SB179M | Guanine nucleotide-binding protein G(q) subunit alpha | Regulator of G-protein signaling 2 | 23434405 | IC50=0.27 ± 0.06 uM
LogEC50 (n)=2.1 ± 0.03 nM (20) | IC50=0.13 ± 0.03 uM
Log EC50 (n)=1.7 ± 0.09 nM (5) | flow-cytometry-based assay，25°C |
| 4EKC_A_B | SB179N | Guanine nucleotide-binding protein G(q) subunit alpha | Regulator of G-protein signaling 2 | 23434405 | IC50=0.27 ± 0.06 uM
LogEC50 (n)=2.1 ± 0.03 nM (20) | IC50=0.69 ± 0.1 uM
Log EC50 (n)=2.3 ± 0.06 nM (7) | flow-cytometry-based assay，25°C |
| 4EKC_A_B | EB182A | Guanine nucleotide-binding protein G(q) subunit alpha | Regulator of G-protein signaling 2 | 23434405 | IC50=0.27 ± 0.06 uM
LogEC50 (n)=2.1 ± 0.03 nM (20) | IC50=0.30 ± 0.04 uM
Log EC50 (n)=2.2 ± 0.05 nM (4) | flow-cytometry-based assay，25°C |
| 4EKC_A_B | NB183A | Guanine nucleotide-binding protein G(q) subunit alpha | Regulator of G-protein signaling 2 | 23434405 | IC50=0.27 ± 0.06 uM
LogEC50 (n)=2.1 ± 0.03 nM (20) | IC50=1.5 ± 0.2 uM
Log EC50 (n)=2.3 ± 0.03 nM (4) | flow-cytometry-based assay，25°C |
| 4EKC_A_B | NB183F | Guanine nucleotide-binding protein G(q) subunit alpha | Regulator of G-protein signaling 2 | 23434405 | IC50=0.27 ± 0.06 uM
LogEC50 (n)=2.1 ± 0.03 nM (20) | IC50=0.17 ± 0.03 uM
Log EC50 (n)=0.9 ± 0.04 nM (5) | flow-cytometry-based assay，25°C |
| 4EKC_A_B | NB183K | Guanine nucleotide-binding protein G(q) subunit alpha | Regulator of G-protein signaling 2 | 23434405 | IC50=0.27 ± 0.06 uM
LogEC50 (n)=2.1 ± 0.03 nM (20) | IC50=7.1 ± 1 uM
Log EC50 (n)=3.0 ± 0.03 nM (4) | flow-cytometry-based assay，25°C |
| 4EKC_A_B | RA183C/LA78V | Guanine nucleotide-binding protein G(q) subunit alpha | Regulator of G-protein signaling 2 | 23434405 | IC50=0.27 ± 0.06 uM
LogEC50 (n)=2.1 ± 0.03 nM (20) | Log EC50 (n)=2.2 ± 0.05 nM (9) | flow-cytometry-based assay，25°C |
| 4EKC_A_B | RA183C/QA81S | Guanine nucleotide-binding protein G(q) subunit alpha | Regulator of G-protein signaling 2 | 23434405 | IC50=0.27 ± 0.06 uM
LogEC50 (n)=2.1 ± 0.03 nM (20) | Log EC50 (n)=2.4 ± 0.04 nM (4) | flow-cytometry-based assay，25°C |
